Palladium-catalyzed tandem C-H functionalization/cyclization strategy for the synthesis of 5-hydroxybenzofuran derivatives

Sachin S. Ichake, Ashok Konala, Veerababurao Kavala, Chun Wei Kuo, Ching Fa Yao*

*此作品的通信作者

研究成果: 雜誌貢獻期刊論文同行評審

20 引文 斯高帕斯(Scopus)

摘要

A palladium-catalyzed benzoquinone C-H functionalization/ cyclization strategy with terminal alkynes was employed for the synthesis of some biologically relevant 2, 3-disubstituted 5-hydroxybenzofuran derivatives. The benzoquinone acts as a reactant as well as an oxidant. During the process, an additional alkyne functionality can be introduced at the C3 position of the benzofuran. Base, ligand, and external oxidant are not required in this protocol.

原文英語
頁(從 - 到)54-57
頁數4
期刊Organic Letters
19
發行號1
DOIs
出版狀態已發佈 - 2017 一月 6

ASJC Scopus subject areas

  • 生物化學
  • 物理與理論化學
  • 有機化學

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