Abstract
An efficient synthesis of functionalized benzofurans is achieved under mild and metal-free conditions from stable para-quinone methides by treatment with phosphine, acyl chloride, and a base. This one-pot phospha-1,6-addition/O-acylation/Wittig reaction is also demonstrated under catalytic conditions with similar efficacy.
| Original language | English |
|---|---|
| Pages (from-to) | 8008-8012 |
| Number of pages | 5 |
| Journal | Organic Letters |
| Volume | 21 |
| Issue number | 19 |
| DOIs | |
| Publication status | Published - 2019 Oct 4 |
ASJC Scopus subject areas
- Biochemistry
- Physical and Theoretical Chemistry
- Organic Chemistry
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CCDC 1952659: Experimental Crystal Structure Determination
Liou, Y.-C. (Contributor), Karanam, P. (Contributor), Jang, Y.-J. (Contributor) & Lin, W. (Contributor), Unknown Publisher, 2019
DOI: 10.5517/ccdc.csd.cc23jx0l, http://www.ccdc.cam.ac.uk/services/structure_request?id=doi:10.5517/ccdc.csd.cc23jx0l&sid=DataCite
Dataset
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CCDC 1943703: Experimental Crystal Structure Determination
Liou, Y.-C. (Contributor), Karanam, P. (Contributor), Jang, Y.-J. (Contributor) & Lin, W. (Contributor), Unknown Publisher, 2019
DOI: 10.5517/ccdc.csd.cc237l32, http://www.ccdc.cam.ac.uk/services/structure_request?id=doi:10.5517/ccdc.csd.cc237l32&sid=DataCite
Dataset